Search Result "3-d]pyrimidine derivatives"


Review Article

The Application of Pyrrolo[2, 3-d]pyrimidine Scaffold in Medicinal Chemistryfrom 2017 to 2021

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 23 Issue: 10 Year: 2023 Page: 1118-1136
Author(s):

An Efficiently Sonochemical Synthesis of Novel Pyrazoles, Bipyrazoles and Pyrazol-3- ylPyrazolo[3,4-d]pyrimidines Incorporating 1H-benzoimidazole Moiety

Journal: Current Organic Chemistry
Volume: 17 Issue: 2 Year: 2013 Page: 194-202
Author(s): Nesreen S. Ahmed,Tamer S. Saleh,El-Sayed H. El-Mossalamy

Research Article

Synthesis, Docking Study of Some Novel Chromeno[4',3'-b]Pyrano[6,5-d]Pyrimidine Derivatives Against COVID-19 Main Protease (Mpro) (6LU7, 6M03)

Journal: Current Computer-Aided Drug Design
Volume: 20 Issue: 5 Year: 2024 Page: 551-563
Author(s): Zahra Rostami Ghalhar

Research Article

Synthesis and Preliminarily Cytotoxicity to A549, HCT116 and MCF-7 Cell Lines of thieno[2,3-d]pyrimidine Derivatives Containing Isoxazole Moiety

Journal: Letters in Drug Design & Discovery
Volume: 15 Issue: 5 Year: 2018 Page: 463-474
Author(s): Jianping Yong,Canzhong Lu,Xiaoyuan Wu

Research Article

Synthesis and Evaluation of Antimicrobial Activity and Molecular Docking of New N-1,3-thiazol-2-ylacetamides of Condensed Pyrido[3',2':4,5] furo(thieno)[3,2-d]pyrimidines

Journal: Current Topics in Medicinal Chemistry
Volume: 20 Issue: 2 Year: 2020 Page: 2192-2209
Author(s): S.N. Sirakanyan,V.G. Kartsev,A. Geronikaki,D. Spinelli,A. Petrou,E.K. Hakobyan,J. Glamoclij,M. Ivanov,M. Sokovic,A.A. Hovakimyan

Synthesis of Novel Derivatives of pyrano[2,3-d]pyrimidinevia Intramolecular Cyclocondensation Reaction Under Acidic and Basic Conditions

Journal: Letters in Organic Chemistry
Volume: 9 Issue: 6 Year: 2012 Page: 386-389
Author(s): Ahmed Al-Sheikh,Kamal Sweidan,Munjed Ibrahim,Mohammed Alarjah,Norbert Kuhn

Research Article

In silico Analysis and Molecular Docking Studies of Novel 4-Amino-3- (Isoquinolin-4-yl)-1H-Pyrazolo[3,4-d]Pyrimidine Derivatives as Dual PI3-K/mTOR Inhibitors

Journal: Current Drug Discovery Technologies
Volume: 16 Issue: 3 Year: 2019 Page: 297-306
Author(s): Ishan I. Panchal,Sandip N. Badeliya,Rakesh Patel,Ashish Patel,Animesh Devaligar

Synthesis and Antioxidant Activity of 1,2,4-Triazole linked Thieno[2,3- d]pyrimidine Derivatives

Journal: Letters in Drug Design & Discovery
Volume: 10 Issue: 2 Year: 2013 Page: 186-193
Author(s): Suresh Maddila,Avula S. Kumar,Sridevi Gorle,M. Singh,Palakondu Lavanya,S.B. Jonnalagadda

Research Article

Novel 1,2,3-Triazole-functionalized pyrido[3',2':4,5]furo[3,2-d]pyrimidin- 4(3H)-one Derivatives: Synthesis, Anticancer Activity, CoMFA and CoMSIA Studies

Journal: Letters in Organic Chemistry
Volume: 17 Issue: 1 Year: 2020 Page: 969-978
Author(s): Sailu Betala,Balakishan Vadla

Research Article

Synthesis and Molecular Docking of New Thiophene Derivatives as Lactate Dehydrogenase-A Inhibitors

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 19 Issue: 1 Year: 2019 Page: 833-841
Author(s): Abd El-Galil E. Amr,Mohamed F. El-Shehry,Alhussein A. Ibrahim,Hanaa M. Hosni,Mohamed A. Al-Omar,Hazem A. Ghabbour

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